Compile Data Set for Download or QSAR
Found 70 of ki data for polymerid = 50004854
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279715(CHEMBL4162544)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279757(CHEMBL4166160)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279763(CHEMBL4162308)copy SMILEScopy InChI
Affinity DataKi: <1.30nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279744(CHEMBL4165984)copy SMILEScopy InChI
Affinity DataKi: <2nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279773(CHEMBL4173915)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279743(CHEMBL4170479)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279720(CHEMBL4177229)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279737(CHEMBL4170653)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279734(CHEMBL4177445)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279723(CHEMBL4165949)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279759(CHEMBL4172982)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279736(CHEMBL4162511)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279748(CHEMBL4170446)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279751(CHEMBL4162719)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of human plasma renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279750(CHEMBL4159344)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279746(CHEMBL4169382)copy SMILEScopy InChI
Affinity DataKi:  38nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279733(CHEMBL4174082)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279742(CHEMBL4166840)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279735(CHEMBL4173877)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279777(CHEMBL4172772)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279781(CHEMBL4162101)copy SMILEScopy InChI
Affinity DataKi:  72nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279802(CHEMBL4159392)copy SMILEScopy InChI
Affinity DataKi:  81nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279793(CHEMBL4174513)copy SMILEScopy InChI
Affinity DataKi:  82nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279724(CHEMBL4167265)copy SMILEScopy InChI
Affinity DataKi:  88nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279722(CHEMBL4170024)copy SMILEScopy InChI
Affinity DataKi:  98nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279786(CHEMBL4166603)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279785(CHEMBL4176818)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279799(CHEMBL4164081)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279930(CHEMBL4173464)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279721(CHEMBL4162756)copy SMILEScopy InChI
Affinity DataKi:  230nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421673(CHEMBL5283441)copy SMILEScopy InChI
Affinity DataKi:  290nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279857(CHEMBL4176150)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279783(CHEMBL4164260)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421686(CHEMBL5282194)copy SMILEScopy InChI
Affinity DataKi:  320nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50293150(CHEMBL468963 | D3RKN_26 | GSK screening, 38 | N-(4...)copy SMILEScopy InChI
Affinity DataKi:  420nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421679(CHEMBL5282708)copy SMILEScopy InChI
Affinity DataKi:  440nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421671(CHEMBL5266831)copy SMILEScopy InChI
Affinity DataKi:  470nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421672(CHEMBL5316225)copy SMILEScopy InChI
Affinity DataKi:  580nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421685(CHEMBL5280226)copy SMILEScopy InChI
Affinity DataKi:  700nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279745(CHEMBL4166200)copy SMILEScopy InChI
Affinity DataKi:  960nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (M1 to G279 residues) expressed in Escherichia coli BL21 (DE3) cells using [T-33P]ATP as substrate afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421687(CHEMBL5277580)copy SMILEScopy InChI
Affinity DataKi:  970nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279841(CHEMBL4174912)copy SMILEScopy InChI
Affinity DataKi:  990nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421681(CHEMBL5273566)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421683(CHEMBL5283041)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421676(CHEMBL5283475)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50279782(CHEMBL4165542)copy SMILEScopy InChI
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of HMG-CoA reductase in rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2183910PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421680(CHEMBL5277737)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421682(CHEMBL5285809)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421684(CHEMBL5277619)copy SMILEScopy InChI
Affinity DataKi:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Vertex Pharmaceuticals Inc

Curated by ChEMBL
LigandPNGBDBM50421674(CHEMBL5284844)copy SMILEScopy InChI
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails
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